Structure-based design, synthesis and biological evaluation of novel ß-secretase inhibitors containing a pyrazole or thiazole moiety as the P3 ligand.
Ghosh, Arun K; Brindisi, Margherita; Yen, Yu-Chen; Xu, Xiaoming; Huang, Xiangping; Devasamudram, Thippeswamy; Bilcer, Geoffrey; Lei, Hui; Koelsch, Gerald; Mesecar, Andrew D; Tang, Jordan.
Bioorg Med Chem Lett
; 25(3): 668-72, 2015 Feb 01.
Artigo em Inglês | MEDLINE | ID: mdl-25537272
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