Structure-activity relationship in the 3-iodo-4-phenoxypyridinone (IOPY) series: The nature of the C-3 substituent on anti-HIV activity.
Benjahad, Abdellah; Oumouch, Said; Guillemont, Jerôme; Pasquier, Elisabeth; Mabire, Dominique; Andries, Koen; Nguyen, Chi Hung; Grierson, David S.
Bioorg Med Chem Lett
; 17(3): 712-6, 2007 Feb 01.
Artigo em Inglês | MEDLINE | ID: mdl-17157017
Design, synthesis and biological evaluation of novel acetamide-substituted doravirine and its prodrugs as potent HIV-1 NNRTIs.
Discovery of 2-pyridone derivatives as potent HIV-1 NNRTIs using molecular hybridization based on crystallographic overlays.
CD8(+) T Cells and cART: A Dynamic Duo?
Design, Synthesis and In Vitro Evaluation of Novel Anti-HIV 3-Pyrazol-3- yl-Pyridin-2-One Analogs.
Focus on Chirality of HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors.
Synthesis and evaluation of pyridinium polyoxometalates as anti-HIV-1 agents.
Synthesis and Anti-HIV Activity of Guanine Modified Fluorinated Acyclic Nucleoside Phosphonate Derivatives.
Microwave-Assisted Expeditious Synthesis of 2-Alkyl-2-(<i>N</i>-arylsulfonylindol-3-yl)-3-<i>N</i>-acyl-5-aryl-1,3,4-oxadiazolines Catalyzed by HgCl2 under Solvent-Free Conditions as Potential Anti-HIV-1 Agents.
Design, synthesis and anti-HIV-1 evaluation of hydrazide-based peptidomimetics as selective gelatinase inhibitors.
<i>In Vitro</i> Antiviral Activity of Cabotegravir against HIV-2.