Synthesis and structure-activity relationships of 1,2,3,4-tetrahydropyrido[2,3-b]pyrazines as potent and selective inhibitors of the anaplastic lymphoma kinase.
Milkiewicz, Karen L; Weinberg, Linda R; Albom, Mark S; Angeles, Thelma S; Cheng, Mangeng; Ghose, Arup K; Roemmele, Renee C; Theroff, Jay P; Underiner, Ted L; Zificsak, Craig A; Dorsey, Bruce D.
Bioorg Med Chem
; 18(12): 4351-62, 2010 Jun 15.
Artigo em Inglês | MEDLINE | ID: mdl-20483621
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